Halogen exchange (Halex) reaction of 5-iodo-1,2,3-triazoles: Synthesis and applications of 5-fluorotriazoles

Brady T. Worrell, Jason E. Hein, Valery V. Fokin

Результат исследований: Материалы для журналаСтатья

53 Цитирования (Scopus)

Выдержка

A good exchange: 5-Iodo-1,2,3-triazoles undergo facile substitution reactions with fluoride salts, thus providing ready access to 5-fluorotriazoles (see scheme). The latter can be further elaborated with various nucleophiles to furnish fully substituted 1,2,3-triazole compounds.

Язык оригиналаАнглийский
Страницы (с-по)11791-11794
Число страниц4
ЖурналAngewandte Chemie - International Edition
Том51
Номер выпуска47
DOI
СостояниеОпубликовано - 19 ноя 2012
Опубликовано для внешнего пользованияДа

Отпечаток

Nucleophiles
Halogens
Triazoles
Fluorides
Ion exchange
Substitution reactions
Salts
5-iodo-1,2,3-triazole

ASJC Scopus subject areas

  • Chemistry(all)
  • Catalysis

Цитировать

Halogen exchange (Halex) reaction of 5-iodo-1,2,3-triazoles : Synthesis and applications of 5-fluorotriazoles. / Worrell, Brady T.; Hein, Jason E.; Fokin, Valery V.

В: Angewandte Chemie - International Edition, Том 51, № 47, 19.11.2012, стр. 11791-11794.

Результат исследований: Материалы для журналаСтатья

Worrell, Brady T. ; Hein, Jason E. ; Fokin, Valery V. / Halogen exchange (Halex) reaction of 5-iodo-1,2,3-triazoles : Synthesis and applications of 5-fluorotriazoles. В: Angewandte Chemie - International Edition. 2012 ; Том 51, № 47. стр. 11791-11794.
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