Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited

Antoni Krasiński, Valery V. Fokin, K. Barry Sharpless

Результат исследований: Материалы для журналаСтатья

212 Цитирования (Scopus)

Выдержка

After revisiting earlier works reporting the regioselective synthesis of 1,5-disubstituted-1,2,3-triazoles via the addition of bromomagnesium acetylides to azides, much improved yields of the products were obtained for a wide array of azides and alkynes. The intermediates of that reaction can be trapped with different electrophiles to regioselectively form 1,4,5-trisubstituted 1,2,3-triazoles.

Язык оригиналаАнглийский
Страницы (с-по)1237-1240
Число страниц4
ЖурналOrganic Letters
Том6
Номер выпуска8
DOI
СостояниеОпубликовано - 15 апр 2004
Опубликовано для внешнего пользованияДа

Отпечаток

Triazoles
Azides
alkynes
Alkynes
synthesis
products

ASJC Scopus subject areas

  • Molecular Medicine

Цитировать

Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. / Krasiński, Antoni; Fokin, Valery V.; Sharpless, K. Barry.

В: Organic Letters, Том 6, № 8, 15.04.2004, стр. 1237-1240.

Результат исследований: Материалы для журналаСтатья

Krasiński, A, Fokin, VV & Sharpless, KB 2004, 'Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited', Organic Letters, том. 6, № 8, стр. 1237-1240. https://doi.org/10.1021/ol0499203
Krasiński, Antoni ; Fokin, Valery V. ; Sharpless, K. Barry. / Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. В: Organic Letters. 2004 ; Том 6, № 8. стр. 1237-1240.
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