• 877 Citations
  • 16 h-Index
1986 …2019
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  • 1 Similar Profiles
Formyl Peptide Receptor Medicine & Life Sciences
Secretory Proteinase Inhibitory Proteins Medicine & Life Sciences
Quantitative Structure-Activity Relationship Medicine & Life Sciences
Derivatives Chemical Compounds
Leukocyte Elastase Medicine & Life Sciences
Molecular modeling Chemical Compounds
Molecules Chemical Compounds
Structure-Activity Relationship Medicine & Life Sciences

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Research Output 1986 2019

  • 877 Citations
  • 16 h-Index
  • 62 Article
  • 5 Conference contribution
  • 3 Review article
  • 1 Comment/debate

Further modifications of 1H-pyrrolo[2,3-b]pyridine derivatives as inhibitors of human neutrophil elastase

Giovannoni, M. P., Cantini, N., Crocetti, L., Guerrini, G., Iacovone, A., Schepetkin, I. A., Vergelli, C., Khlebnikov, A. I. & Quinn, M. T., 1 Jan 2019, In : Drug Development Research.

Research output: Contribution to journalArticle

Secretory Proteinase Inhibitory Proteins
Leukocyte Elastase
Multifunctional Enzymes
pyrrolo(2, 3-b)pyridine
Respiratory System
1 Citation (Scopus)

Inhibition of T Cell Receptor Activation by Semi-Synthetic Sesquiterpene Lactone Derivatives and Molecular Modeling of Their Interaction with Glutathione and Tyrosine Kinase ZAP-70

Khlebnikov, A. I., Schepetkin, I. A., Kishkentaeva, A. S., Shaimerdenova, Z. R., Atazhanova, G. A., Adekenov, S. M., Kirpotina, L. N. & Quinn, M. T., 19 Jan 2019, In : Molecules (Basel, Switzerland). 24, 2

Research output: Contribution to journalArticle

glutathione
Molecular modeling
Sesquiterpenes
tyrosine
Lactones

Synthesis, biological evaluation, and molecular modeling of 11H-indeno[1,2-b]quinoxalin-11-one derivatives and tryptanthrin-6-oxime as c-Jun N-terminal kinase inhibitors

Schepetkin, I. A., Khlebnikov, A. I., Potapov, A. S., Kovrizhina, A. R., Matveevskaya, V. V., Belyanin, M. L., Atochin, D. N., Zanoza, S. O., Gaidarzhy, N. M., Lyakhov, S. A., Kirpotina, L. N. & Quinn, M. T., 1 Jan 2019, In : European Journal of Medicinal Chemistry. 161, p. 179-191 13 p.

Research output: Contribution to journalArticle

Quinoxalines
Molecular modeling
Oximes
JNK Mitogen-Activated Protein Kinases
Derivatives
2 Citations (Scopus)

1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitors

Crocetti, L., Giovannoni, M. P., Schepetkin, I. A., Quinn, M. T., Khlebnikov, A. I., Cantini, N., Guerrini, G., Iacovone, A., Teodori, E. & Vergelli, C., 15 Nov 2018, In : Bioorganic and Medicinal Chemistry. 26, 21, p. 5583-5595 13 p.

Research output: Contribution to journalArticle

Secretory Proteinase Inhibitory Proteins
Leukocyte Elastase
Scaffolds
Indazoles
Oxadiazoles
2 Citations (Scopus)

4-Aroyl-3-hydroxy-5-phenyl-1H-pyrrol-2(5H)-ones as N-formyl peptide receptor 1 (FPR1) antagonists

Kirpotina, L. N., Schepetkin, I. A., Khlebnikov, A. I., Ruban, O. I., Ge, Y., Ye, R. D., Kominsky, D. J. & Quinn, M. T., 2017, (Accepted/In press) In : Biochemical Pharmacology. 142, p. 120-132 13 p.

Research output: Contribution to journalArticle

Formyl Peptide Receptor
HL-60 Cells
Pyrroles
Neutrophils
Trp-Lys-Tyr-Met-Val-Met